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Review article

The role of ligand efficiency metrics in drug discovery

Andrew L. HopkinsDivision of Biological Chemistry and Drug Discovery, College of Life Sciences, University of Dundee, Dundee DD1 5EH, UKGyörgy M. KeserűResearch Centre for Natural Sciences, Hungarian Academy of Sciences, 1117 Budapest, Magyar Tudósok körútja 2., 1525 Budapest, PO Box 17, HungaryPaul D. LeesonGlaxoSmithKline, Medicines Research Centre, Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, UKDavid C. ReesCharles H. ReynoldsGfree Bio, 3805 Old Easton Road, Doylestown, Pennsylvania 18902, USA
2014en
ABI

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Cited by 50 references