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Synthesis, anticancer activity and molecular modeling studies of 1,2,4-triazole derivatives as EGFR inhibitors

Hany A.M. El-SheriefDepartment of Pharmaceutical Chemistry, Faculty of Pharmacy, Nahda University, Beni-suef, Egypt; Department of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, Aljouf, Sakaka, 2014, Saudi Arabia. Electronic address: [email protected]Bahaa G. M. YoussifDepartment of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Assiut University, Assiut, 71526, Egypt; Department of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, Aljouf, Sakaka, 2014, Saudi ArabiaSyed Nasir Abbas BukhariDepartment of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, Aljouf, Sakaka, 2014, Saudi ArabiaAhmed H. AbdelazeemDepartment of Medicinal Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, 62514, EgyptMohamed Abdel‐AzizDepartment of Medicinal Chemistry, Faculty of Pharmacy, Minia University, 61519, Minia, Egypt. Electronic address: [email protected]Hamdy M. Abdel‐RahmanDepartment of Pharmaceutical Chemistry, Faculty of Pharmacy, Nahda University, Beni-suef, Egypt; Department of Medicinal Chemistry, Faculty of Pharmacy, Assiut University, 71526, Assiut, Egypt
2018en
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