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Synthesis and structure–activity relationships of potent and orally active sulfonamide ETB selective antagonists

Yasuhiko KandaShionogi Research Laboratories, Shionogi & Co, Ltd, Osaka, Japan. [email protected]Yasuyuki KawanishiShionogi Research Laboratories, Shionogi & Co., Ltd., Fukushima-ku, Osaka 553–0002, JapanKatsuo OdaShionogi Research Laboratories, Shionogi & Co., Ltd., Fukushima-ku, Osaka 553–0002, JapanTeruo SakataShionogi Research Laboratories, Shionogi & Co., Ltd., Fukushima-ku, Osaka 553–0002, JapanShin‐ichi MiharaShionogi Research Laboratories, Shionogi & Co., Ltd., Fukushima-ku, Osaka 553–0002, JapanKenji AsakuraShionogi Research Laboratories, Shionogi & Co., Ltd., Toyonaka, Osaka 561–0825, JapanToshiyuki KanemasaShionogi Research Laboratories, Shionogi & Co., Ltd., Toyonaka, Osaka 561–0825, JapanMitsuyoshi NinomiyaShionogi Research Laboratories, Shionogi & Co., Ltd., Toyonaka, Osaka 561–0825, JapanMasafumi FujimotoShionogi Research Laboratories, Shionogi & Co., Ltd., Fukushima-ku, Osaka 553–0002, JapanToshiro KonoikeShionogi Research Laboratories, Shionogi & Co., Ltd., Amagasaki, Hyogo 660–0813, Japan
2001en
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